GHRP-6
Growth Hormone Releasing Peptide 6
Evidence & Status
- Preliminary / Experimental
- Preliminary
At a Glance
A growth hormone-releasing peptide studied for its ability to stimulate growth hormone secretion and, notably, to strongly stimulate appetite — a property that has attracted research interest in muscle wasting and cachexia contexts.
Plain English
Researchers study GHRP-6 because it acts on the ghrelin receptor to stimulate growth hormone release and also produces a significant increase in appetite. Scientists are particularly interested in the appetite-stimulating mechanism as it relates to conditions where loss of appetite and muscle mass is a serious concern, such as cancer-related cachexia or severe illness. It is one of the earlier growth hormone secretagogues and has contributed significantly to scientific understanding of how ghrelin receptors function.
Overview
An early synthetic growth-hormone-releasing hexapeptide studied in experimental human and animal research. It is not FDA-approved, and its short-term pharmacodynamic effects do not establish clinical benefit or a treatment regimen.
Research Summary
Experimental studies in healthy men found that the GHRP-6 sequence can stimulate growth-hormone secretion, and preclinical work supports a receptor mechanism distinct from GHRH. These observations are historical and mechanistic; they do not establish clinical efficacy, long-term safety, or a use protocol.
Research Areas
- GH release
- Appetite stimulation & cachexia
- Muscle wasting
- Wound healing
- Cardioprotection
Safety & Risks
Serious Risks
- Experimental endocrine and appetite effects have been reported; long-term safety and clinical outcomes have not been established
Reported Side Effects
- Significant hunger increase (most common)
- Cortisol elevation
- Prolactin increase
- Water retention
- Fatigue
Legal Status by Region
- United States
- Research only
- United Kingdom
- Research only
- Australia
- Research only
- Canada
- Research only
Citations & Sources
- Oral administration of growth hormone (GH)-releasing peptide stimulates GH secretion in normal men
Journal of Clinical Endocrinology & Metabolism · 1992
PMID 1592884
- Desensitization studies using perifused rat pituitary cells show that growth hormone-releasing hormone and His-D-Trp-Ala-Trp-D-Phe-Lys-NH2 stimulate growth hormone release through distinct receptor sites
1991
PMID 1674284
- Twenty-four-hour growth hormone (GH)-releasing peptide (GHRP) infusion enhances pulsatile GH secretion and specifically attenuates the response to a subsequent GHRP bolus
Huhn WC, Hartman ML, Pezzoli SS, Thorner MO · Journal of Clinical Endocrinology and Metabolism · 1993
PMID 8496311 · DOI 10.1210/jcem.76.5.8496311