P021
P021 (CNTF-derived neurotrophic research peptide)
Evidence & Status
- Preliminary / Experimental
- Preliminary
At a Glance
A modified CNTF-derived pentapeptide studied only in verified animal models. It has no verified human interventional evidence, established human pharmacokinetics, or established human safety profile.
Plain English
Researchers study the exact modified P021 construct in animal models. These findings do not establish human neurogenesis, clinical benefit, pharmacokinetics, safety, or a treatment protocol.
Overview
P021 is a modified CNTF-derived pentapeptide, Ac-DGGL(A)G-NH2, in which the adamantyl group modifies the C-terminal glycine rather than adding a sixth amino-acid residue. The approved evidence concerns chronic oral treatment in mouse models; it does not establish human pharmacokinetics, clinical efficacy, or dosing.
Research Summary
Two approved publications report P021 in transgenic mouse models of Alzheimer's disease–related pathology. These are preclinical findings from a limited evidence base and must not be converted into claims of human neurogenesis, cognitive benefit, safety, or a treatment protocol.
Research Areas
- Hippocampal neurogenesis
- Cognitive aging
- Alzheimer's disease
- CNTF signaling pathway
- Synaptic plasticity
Safety & Risks
Serious Risks
- Complete absence of human safety data
- Unknown CNS effects at non-physiological concentrations
- Theoretical risk of aberrant neurogenesis or gliosis at supratherapeutic doses
- Field of adult human hippocampal neurogenesis itself is scientifically contested
Reported Side Effects
- Unknown in humans
Legal Status by Region
- United States
- The cited evidence is preclinical and does not establish regulatory authorization or a human clinical indication.
- United Kingdom
- The cited evidence is preclinical and does not establish regulatory authorization or a human clinical indication.
- Australia
- The cited evidence is preclinical and does not establish regulatory authorization or a human clinical indication.
- Canada
- The cited evidence is preclinical and does not establish regulatory authorization or a human clinical indication.
Citations & Sources
- Disease modifying effect of chronic oral treatment with a neurotrophic peptidergic compound in a triple transgenic mouse model of Alzheimer's disease.
Kazim SF et al. · Neurobiology of Disease · 2014
PMID 25046994 · DOI 10.1016/j.nbd.2014.07.001
- Prevention of dendritic and synaptic deficits and cognitive impairment with a neurotrophic compound.
Baazaoui N, Iqbal K · Alzheimer's Research & Therapy · 2017
PMID 28655344 · DOI 10.1186/s13195-017-0273-7